Description
Latin name
Clenbuterol
Release form
Tablets.
Packaging
A carton pack contains 50 tablets.
Pharmacological action
Clenbuterol is a selective 2-adrenergic agonist. It has a bronchodilator and secretolytic effect. It excites 2-adrenergic receptors, stimulates adenylate cyclase, increases the content of cAMP in the cells, which, affecting the protein kinase system, deprives myosin of the ability to bind to actin and promotes relaxation of the bronchi. It inhibits the release of mediators from mast cells that contribute to bronchospasm and inflammation of the bronchi. Reduces edema or congestion in the bronchi, improves mucociliary clearance.
Indications
Bronchial asthma, chronic obstructive pulmonary disease.
Contraindications
Contraindicated in pregnancy and lactation.
Use during pregnancy and lactation
Use is prohibited.
Composition
Active ingredient: Clenbuterol hydrochloride – 5 mcg.
Excipients: lactose monohydrate – 70 mg wheat starch – 31.48 mg MCC – 48, 5 mg silicon colloidal dioxide – 2 mg magnesium stearate – 2 mg povidone (povidone K25) – 6 mg
Dosage and administration
Applied orally.
Adults and children over 12 years old – 10–20 mcg 2-3 times a day, maintenance dose – 10 mcg 2 times a day.
Young children – in reduced doses, depending on age, 2 times a day.
Side effects of
From the cardiovascular system: tachycardia, extrasystole, arterial hypo- or (more often) hypertension, cardialgia, facial flushing.
From the side of the central nervous system and peripheral nervous system: tremor of fingers, anxiety, headache, dizziness, general weakness, insomnia, paresthesia.
From the digestive system: dry mouth, nausea, vomiting, gastralgia.
Allergic reactions: skin rash, urticaria, bronchospasm, angioedema.
Other: increased sweating, hypokalemia, muscle cramps. With a sharp withdrawal of the drug, the development of resistance and rebound syndrome is possible. When used in large doses, causes tremor of the fingers.
Overdose
Symptoms: arrhythmia, tachycardia, arterial hypertension, cardialgia, tremor of the extremities, hypokalemia may develop.
Treatment: gastric lavage, administration of activated carbon, the use of water-salt solutions, monitoring the level of potassium in the blood serum, symptomatic therapy.
Storage Conditions
List B. The product should be stored in a dark place out of the reach of children at a temperature not exceeding 25 °, and should not be frozen.
Expiration
3 years.
Do not use after the expiry date stated on the package.
active substance
Clenbuterol
Terms leave around drugstore
prescription
lekarstvennaja form
tablets
Prescribing rdlkp Adults prescribed by a doctor
Sofarma Bolgaria
